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  Bacterial Infections and Mycoses

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Articles published in J Med Chem

Retrieve available abstracts of 35 articles:
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Single Articles


    December 2017
  1. GUAN D, Chen F, Xiong L, Tang F, et al
    Extra sugar on vancomycin: new analogues for combating multidrug-resistant Staphylococcus aureus and vancomycin-resistant Enterococci.
    J Med Chem. 2017 Dec 15. doi: 10.1021/acs.jmedchem.7b01345.
    PubMed     Text format     Abstract available


  2. CAMERON AJ, Edwards PJB, Harjes E, Sarojini V, et al
    Tyrocidine A Analogues Bearing the Planar d-Phe-2-Abz Turn Motif: How Conformation Impacts Bioactivity.
    J Med Chem. 2017;60:9565-9574.
    PubMed     Text format     Abstract available


  3. MOON SH, Zhang X, Zheng G, Meeker DG, et al
    Novel Linear Lipopeptide Paenipeptins with Potential for Eradicating Biofilms and Sensitizing Gram-Negative Bacteria to Rifampicin and Clarithromycin.
    J Med Chem. 2017;60:9630-9640.
    PubMed     Text format     Abstract available


  4. CHOI H, Ham SY, Cha E, Shin Y, et al
    Structure-Activity Relationships of 6- and 8-Gingerol Analogs as Anti-Biofilm Agents.
    J Med Chem. 2017;60:9821-9837.
    PubMed     Text format     Abstract available


    October 2017
  5. GOOD JAD, Kulen M, Silver J, Krishnan KS, et al
    Thiazolino 2-pyridone amide isosteres as inhibitors of Chlamydia trachomatis infectivity.
    J Med Chem. 2017 Oct 20. doi: 10.1021/acs.jmedchem.7b00716.
    PubMed     Text format     Abstract available


    September 2017
  6. LI X, Hernandez V, Rock FL, Choi W, et al
    Discovery of a Potent and Specific M. tuberculosis Leucyl-tRNA Synthetase Inhibitor: (S)-3-(Aminomethyl)-4-chloro-7-(2-hydroxyethoxy)benzo[c][1,2]oxaborol-1(3H)-ol (GSK656).
    J Med Chem. 2017 Sep 27. doi: 10.1021/acs.jmedchem.7b00631.
    PubMed     Text format     Abstract available


  7. BUCHIERI MV, Cimino M, Rebollo-Ramirez S, Beauvineau C, et al
    Nitazoxanide Analogs Require Nitroreduction for Antimicrobial Activity in Mycobacterium smegmatis.
    J Med Chem. 2017;60:7425-7433.
    PubMed     Text format     Abstract available


  8. CHEN AY, Thomas PW, Stewart AC, Bergstrom A, et al
    Dipicolinic Acid Derivatives as Inhibitors of New Delhi Metallo-beta-lactamase-1.
    J Med Chem. 2017;60:7267-7283.
    PubMed     Text format     Abstract available


  9. ABDEL MONAIM SAH, Ramchuran EJ, El-Faham A, Albericio F, et al
    Converting Teixobactin into a Cationic Antimicrobial Peptide (AMP).
    J Med Chem. 2017;60:7476-7482.
    PubMed     Text format     Abstract available


  10. NI S, Wei H, Li B, Chen F, et al
    Novel Inhibitors of Staphyloxanthin Virulence Factor in Comparison with Linezolid and Vancomycin versus Methicillin-Resistant, Linezolid-Resistant and Vancomycin-Intermediate Staphylococcus aureus Infections in vivo.
    J Med Chem. 2017 Sep 7. doi: 10.1021/acs.jmedchem.7b00949.
    PubMed     Text format     Abstract available


    July 2017
  11. KOZIKOWSKI AP, Onajole OK, Stec J, Dupont C, et al
    Targeting Mycolic Acid Transport by Indole-2-carboxamides for the Treatment of Mycobacterium abscessus Infections.
    J Med Chem. 2017;60:5876-5888.
    PubMed     Text format     Abstract available


    June 2017
  12. PIIZZI G, Parker DT, Peng Y, Dobler M, et al
    Design, Synthesis, and Properties of a Potent Inhibitor of Pseudomonas aeruginosa Deacetylase LpxC.
    J Med Chem. 2017;60:5002-5014.
    PubMed     Text format     Abstract available


  13. LIN S, Koh JJ, Aung TT, Sin WLW, et al
    Semisynthetic Flavone-Derived Antimicrobials with Therapeutic Potential against Methicillin-Resistant Staphylococcus aureus (MRSA).
    J Med Chem. 2017 Jun 21. doi: 10.1021/acs.jmedchem.7b00380.
    PubMed     Text format     Abstract available


  14. LIU F, Dawadi S, Maize KM, Dai R, et al
    Structure-Based Optimization of Pyridoxal 5'-Phosphate (PLP)-Dependent Transaminase Enzyme (BioA) Inhibitors that Target Biotin Biosynthesis in Mycobacterium tuberculosis.
    J Med Chem. 2017 Jun 8. doi: 10.1021/acs.jmedchem.7b00189.
    PubMed     Text format     Abstract available


    May 2017
  15. PANCHAUD P, Bruyere T, Blumstein AC, Bur D, et al
    Discovery and Optimization of Isoquinoline Ethyl Ureas as Antibacterial Agents.
    J Med Chem. 2017;60:3755-3775.
    PubMed     Text format     Abstract available


  16. BHOWMICK M, Tokmina-Roszyk D, Onwuha-Ekpete L, Harmon K, et al
    Second Generation Triple-Helical Peptide Inhibitors of Matrix Metalloproteinases.
    J Med Chem. 2017;60:3814-3827.
    PubMed     Text format     Abstract available


  17. MAYER K, Eris D, Schwardt O, Sager CP, et al
    Urinary Tract Infection - Which Conformation of the Bacterial Lectin FimH Is Therapeutically Relevant?
    J Med Chem. 2017 May 4. doi: 10.1021/acs.jmedchem.7b00342.
    PubMed     Text format     Abstract available


    April 2017
  18. HAGRAS M, Mohammad H, Mandour MS, Hegazy YA, et al
    Investigating the Antibacterial Activity of Biphenylthiazoles against Methicillin- and Vancomycin-Resistant Staphylococcus aureus (MRSA and VRSA).
    J Med Chem. 2017 Apr 24. doi: 10.1021/acs.jmedchem.7b00392.
    PubMed     Text format     Abstract available


  19. SIRICILLA S, Mitachi K, Yang J, Eslamimehr S, et al
    A New Combination of a Pleuromutilin Derivative and Doxycycline for Treatment of Multidrug-Resistant Acinetobacter baumannii.
    J Med Chem. 2017;60:2869-2878.
    PubMed     Text format     Abstract available


  20. YANG T, Moreira W, Nyantakyi SA, Chen H, et al
    Amphiphilic Indole Derivatives as Antimycobacterial Agents: Structure-Activity Relationships and Membrane Targeting Properties.
    J Med Chem. 2017;60:2745-2763.
    PubMed     Text format     Abstract available


  21. TAN L, Tao Y, Wang T, Zou F, et al
    Discovery of Novel Pyridone-Conjugated Monosulfactams as Potent and Broad-Spectrum Antibiotics for Multidrug-Resistant Gram-Negative Infections.
    J Med Chem. 2017;60:2669-2684.
    PubMed     Text format     Abstract available


    March 2017
  22. DENG Y, Sun C, Hunt DK, Fyfe C, et al
    Heterocyclyl Tetracyclines. 1. 7-Trifluoromethyl-8-Pyrrolidinyltetracyclines: Potent, Broad Spectrum Antibacterial Agents with Enhanced Activity against Pseudomonas aeruginosa.
    J Med Chem. 2017;60:2498-2512.
    PubMed     Text format     Abstract available


  23. DOU X, Zhu X, Wang J, Dong N, et al
    Novel Design of Heptad Amphiphiles To Enhance Cell Selectivity, Salt Resistance, Antibiofilm Properties and Their Membrane-Disruptive Mechanism.
    J Med Chem. 2017;60:2257-2270.
    PubMed     Text format     Abstract available


  24. HONG WD, Gibbons PD, Leung SC, Amewu R, et al
    Rational Design, Synthesis and Biological Evaluation of Heterocyclic Quinolones Targeting the respiratory chain of Mycobacterium tuberculosis.
    J Med Chem. 2017 Mar 17. doi: 10.1021/acs.jmedchem.6b01718.
    PubMed     Text format     Abstract available


  25. MOHAMMAD H, Younis W, Chen L, Peters CE, et al
    Phenylthiazole Antibacterial Agents Targeting Cell Wall Synthesis Exhibit Potent Activity In Vitro and In Vivo against Vancomycin-resistant Enterococci.
    J Med Chem. 2017 Mar 1. doi: 10.1021/acs.jmedchem.6b01780.
    PubMed     Text format     Abstract available


    February 2017
  26. TOLEDANO-MAGANA Y, Garcia-Ramos JC, Torres-Gutierrez C, Vazquez-Gasser C, et al
    Water-Soluble Ruthenium (II) Chiral Heteroleptic Complexes with Amoebicidal in Vitro and in Vivo Activity.
    J Med Chem. 2017;60:899-912.
    PubMed     Text format     Abstract available


  27. ASTOLFI A, Felicetti T, Iraci N, Manfroni G, et al
    Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors.
    J Med Chem. 2017 Feb 8. doi: 10.1021/acs.jmedchem.6b01439.
    PubMed     Text format     Abstract available


    December 2016
  28. STULAR T, Lesnik S, Rozman K, Schink J, et al
    Discovery of Mycobacterium tuberculosis InhA Inhibitors by Binding Sites Comparison and Ligands Prediction.
    J Med Chem. 2016.
    PubMed     Text format     Abstract available


  29. GARZAN A, Willby MJ, Green KD, Gajadeera CS, et al
    Sulfonamide-Based Inhibitors of Aminoglycoside Acetyltransferase Eis Abolish Resistance to Kanamycin in Mycobacterium tuberculosis.
    J Med Chem. 2016;59:10619-10628.
    PubMed     Text format     Abstract available


    September 2016
  30. GORDON CP, Olson SD, Lister JL, Kavanaugh JS, et al
    Truncated auto-inducing peptides as antagonists of Staphylococcus lugdunensis quorum sensing.
    J Med Chem. 2016.
    PubMed     Text format     Abstract available


    July 2016
  31. BRUNNER K, Maric S, Reshma RS, Almqvist H, et al
    Inhibitors of the cysteine synthase CysM with antibacterial potency against dormant Mycobacterium tuberculosis.
    J Med Chem. 2016.
    PubMed     Text format     Abstract available


    June 2016
  32. PITTA E, Rogacki MK, Balabon O, Huss S, et al
    Searching for new leads for Tuberculosis: Design, synthesis and biological evaluation of novel 2-quinolin-4-yloxyacetamides.
    J Med Chem. 2016.
    PubMed     Text format     Abstract available


  33. BARANOWSKI C, Rubin EJ
    Could Killing Bacterial Subpopulations Hit Tuberculosis out of the Park?
    J Med Chem. 2016.
    PubMed     Text format     Abstract available


  34. STEC J, Onajole OK, Lun S, Guo H, et al
    Indole-2-carboxamide-Based MmpL3 Inhibitors Show Exceptional Antitubercular Activity in an Animal Model of Tuberculosis Infection.
    J Med Chem. 2016.
    PubMed     Text format     Abstract available


    May 2016
  35. YU M, Nagalingam G, Ellis S, Martinez E, et al
    Non-toxic metal-cyclam complexes, a new class of compounds with potency against drug-resistant Mycobacterium tuberculosis.
    J Med Chem. 2016.
    PubMed     Text format     Abstract available


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